百科

(S)-7-((1S,2R)-1,2-bis((4-methoxybenzyl)oxy)-2-(1-methyl-1H-pyrazol-4-yl)ethyl)-3-methyl-6,7-dihydro-4H-[1,2,3]triazolo[5,1-c][1,4]oxazine

(S)-7-((1S,2R)-1,2-bis((4-methoxybenzyl)oxy)-2-(1-methyl-1H-pyrazol-4-yl)ethyl)-3-methyl-6,7-dihydro-4H-[1,2,3]triazolo[5,1-c][1,4]oxazine

CAS号：1442680-72-9

英文名：(S)-7-((1S,2R)-1,2-bis((4-methoxybenzyl)oxy)-2-(1-methyl-1H-pyrazol-4-yl)ethyl)-3-methyl-6,7-dihydro-4H-[1,2,3]triazolo[5,1-c][1,4]oxazine

分子式：C28H33N5O5

分子量：519.592

合成路线

3,4-di-O-(p-methoxybenzyl)-6-O-trityl-D-galactal

3,4-di-O-(p-methoxybenzyl)-6-O-trityl-D-galactal

(S)-7-((1S,2R)-1,2-bis((4-methoxybenzyl)oxy)-2-(1-methyl-1H-pyrazol-4-yl)ethyl)-3-methyl-6,7-dihydro-4H-[1,2,3]triazolo[5,1-c][1,4]oxazine

(S)-7-((1S,2R)-1,2-bis((4-methoxybenzyl)oxy)-2-(1-methyl-1H-pyrazol-4-yl)ethyl)-3-methyl-6,7-dihydro-4H-[1,2,3]triazolo[5,1-c][1,4]oxazine

(2R,3S,4R)-3,4-bis((4-methoxybenzyl)oxy)-4-(1-methyl-1H-pyrazol-4-yl)-1-(trityloxy)butan-2-ol

(2R,3S,4R)-3,4-bis((4-methoxybenzyl)oxy)-4-(1-methyl-1H-pyrazol-4-yl)-1-(trityloxy)butan-2-ol

(S)-7-((1S,2R)-1,2-bis((4-methoxybenzyl)oxy)-2-(1-methyl-1H-pyrazol-4-yl)ethyl)-3-methyl-6,7-dihydro-4H-[1,2,3]triazolo[5,1-c][1,4]oxazine

(S)-7-((1S,2R)-1,2-bis((4-methoxybenzyl)oxy)-2-(1-methyl-1H-pyrazol-4-yl)ethyl)-3-methyl-6,7-dihydro-4H-[1,2,3]triazolo[5,1-c][1,4]oxazine

2-C-formyl-3,4-di-O-(p-methoxybenzyl)-6-O-trityl-D-galactal

2-C-formyl-3,4-di-O-(p-methoxybenzyl)-6-O-trityl-D-galactal

(S)-7-((1S,2R)-1,2-bis((4-methoxybenzyl)oxy)-2-(1-methyl-1H-pyrazol-4-yl)ethyl)-3-methyl-6,7-dihydro-4H-[1,2,3]triazolo[5,1-c][1,4]oxazine

(S)-7-((1S,2R)-1,2-bis((4-methoxybenzyl)oxy)-2-(1-methyl-1H-pyrazol-4-yl)ethyl)-3-methyl-6,7-dihydro-4H-[1,2,3]triazolo[5,1-c][1,4]oxazine

(2R,3R,4R)-2-((trityloxy)methyl)-3,4-dihydro-2H-pyran-3,4-diol

(2R,3R,4R)-2-((trityloxy)methyl)-3,4-dihydro-2H-pyran-3,4-diol

(S)-7-((1S,2R)-1,2-bis((4-methoxybenzyl)oxy)-2-(1-methyl-1H-pyrazol-4-yl)ethyl)-3-methyl-6,7-dihydro-4H-[1,2,3]triazolo[5,1-c][1,4]oxazine

(S)-7-((1S,2R)-1,2-bis((4-methoxybenzyl)oxy)-2-(1-methyl-1H-pyrazol-4-yl)ethyl)-3-methyl-6,7-dihydro-4H-[1,2,3]triazolo[5,1-c][1,4]oxazine

上游原料

2-C-formyl-3,4-di-O-(p-methoxybenzyl)-6-O-trityl-D-galactal 3,4-di-O-(p-methoxybenzyl)-6-O-trityl-D-galactal (2R,3S,4R)-3,4-bis((4-methoxybenzyl)oxy)-4-(1-methyl-1H-pyrazol-4-yl)-1-(trityloxy)butan-2-ol

下游产品

(1R,2S)-1-(1-methyl-1H-pyrazol-4-yl)-2-((S)-3-methyl-6,7-dihydro-4H-[1,2,3]triazolo[5,1-c][1,4]oxazin-7-yl)ethane-1,2-diol