百科

3-{2-[(2S,3R,4R,5S,6S)-6-(5-Azido-pentyloxymethyl)-4-benzyloxy-5-(4-methoxy-benzyloxy)-3-triisopropylsilanyloxy-tetrahydro-pyran-2-yloxy]-ethyl}-1-benzenesulfonyl-1H-indole

3-{2-[(2S,3R,4R,5S,6S)-6-(5-Azido-pentyloxymethyl)-4-benzyloxy-5-(4-methoxy-benzyloxy)-3-triisopropylsilanyloxy-tetrahydro-pyran-2-yloxy]-ethyl}-1-benzenesulfonyl-1H-indole

CAS号：543697-12-7

英文名：3-{2-[(2S,3R,4R,5S,6S)-6-(5-Azido-pentyloxymethyl)-4-benzyloxy-5-(4-methoxy-benzyloxy)-3-triisopropylsilanyloxy-tetrahydro-pyran-2-yloxy]-ethyl}-1-benzenesulfonyl-1H-indole

分子式：C51H68N4O9SSi

分子量：941.258

合成路线

(4aS,6S,7R,8S,8aS)-6-[2-(1-Benzenesulfonyl-1H-indol-3-yl)-ethoxy]-8-benzyloxy-2-(4-methoxy-phenyl)-hexahydro-pyrano[3,2-d][1,3]dioxin-7-ol

(4aS,6S,7R,8S,8aS)-6-[2-(1-Benzenesulfonyl-1H-indol-3-yl)-ethoxy]-8-benzyloxy-2-(4-methoxy-phenyl)-hexahydro-pyrano[3,2-d][1,3]dioxin-7-ol

3-{2-[(2S,3R,4R,5S,6S)-6-(5-Azido-pentyloxymethyl)-4-benzyloxy-5-(4-methoxy-benzyloxy)-3-triisopropylsilanyloxy-tetrahydro-pyran-2-yloxy]-ethyl}-1-benzenesulfonyl-1H-indole

3-{2-[(2S,3R,4R,5S,6S)-6-(5-Azido-pentyloxymethyl)-4-benzyloxy-5-(4-methoxy-benzyloxy)-3-triisopropylsilanyloxy-tetrahydro-pyran-2-yloxy]-ethyl}-1-benzenesulfonyl-1H-indole

(4aS,6S,7S,8S,8aS)-6-[2-(1-Benzenesulfonyl-1H-indol-3-yl)-ethoxy]-8-benzyloxy-2-(4-methoxy-phenyl)-hexahydro-pyrano[3,2-d][1,3]dioxin-7-ol

(4aS,6S,7S,8S,8aS)-6-[2-(1-Benzenesulfonyl-1H-indol-3-yl)-ethoxy]-8-benzyloxy-2-(4-methoxy-phenyl)-hexahydro-pyrano[3,2-d][1,3]dioxin-7-ol

3-{2-[(2S,3R,4R,5S,6S)-6-(5-Azido-pentyloxymethyl)-4-benzyloxy-5-(4-methoxy-benzyloxy)-3-triisopropylsilanyloxy-tetrahydro-pyran-2-yloxy]-ethyl}-1-benzenesulfonyl-1H-indole

3-{2-[(2S,3R,4R,5S,6S)-6-(5-Azido-pentyloxymethyl)-4-benzyloxy-5-(4-methoxy-benzyloxy)-3-triisopropylsilanyloxy-tetrahydro-pyran-2-yloxy]-ethyl}-1-benzenesulfonyl-1H-indole

上游原料

(4aS,6S,7R,8S,8aS)-6-[2-(1-Benzenesulfonyl-1H-indol-3-yl)-ethoxy]-8-benzyloxy-2-(4-methoxy-phenyl)-hexahydro-pyrano[3,2-d][1,3]dioxin-7-ol (4aS,6S,7S,8S,8aS)-6-[2-(1-Benzenesulfonyl-1H-indol-3-yl)-ethoxy]-8-benzyloxy-2-(4-methoxy-phenyl)-hexahydro-pyrano[3,2-d][1,3]dioxin-7-ol

下游产品

5-[(2S,3S,4R,5R,6S)-6-[2-(1-Benzenesulfonyl-1H-indol-3-yl)-ethoxy]-4-benzyloxy-3-(pyridin-3-ylmethoxy)-5-(1-trityl-1H-imidazol-4-ylmethoxy)-tetrahydro-pyran-2-ylmethoxy]-pentylamine (2S,3R,4S,5S,6S)-6-(5-Azido-pentyloxymethyl)-2-[2-(1-benzenesulfonyl-1H-indol-3-yl)-ethoxy]-4-benzyloxy-5-(4-methoxy-benzyloxy)-tetrahydro-pyran-3-ol