(1R,2S)-1-[((1R,4R,5R)-3-oxo-2-oxa-bicyclo[2.2.1]heptane-5-carbonyl)-amino]-2-vinyl-cyclopropane carboxylic acid ethyl ester

(1R,2R,4R)-4-[2-(4-methyl-piperazin-1-yl)-quinazolin-4-yloxy]-cyclopentane-1,2-dicarboxylic acid 1-[((1R,2S)-1-cyclopropanesulfonylaminocarbonyl-2-vinyl-cyclopropyl)amide] 2-(hex-5-enyl-methyl-amide)

(1R,2S)-1-({(1R,2R,4R)-2-(hex-5-enyl-methyl-carbamoyl)-4-[2-(4-isopropyl-thiazol-2-yl)-quinazolin-4-yloxy]-cyclopentanecarbonyl}-amino)-2-vinyl-cyclopropanecarboxylic acid