化合物简介
Regadenoson (CVT-3146, Lexiscan) is an A2A adenosine receptor agonist that is a coronary vasodilator that is commonly used in pharmacologic stress testing. It produces hyperemia quickly and maintains it for a duration that is useful for radionuclide myocardial perfusion imaging. The selective nature of the drug makes it preferable to other stress agents such as adenosine, which are less selective and therefore cause more side-effects.
基本信息
中文名称
瑞加德松
英文名称
Regadenoson
中文别名
2-[4-[(甲基氨基)羰基]-1H-吡唑-1-基]腺苷酸
英文别名
CAS号
313348-27-5
分子式
C15H18N8O5
分子量
390.354
精确质量
390.14
PSA
186.46
LOGP
-1.4626
编号系统
UNII
7AXV542LZ4
物化性质
外观与性状
灰白色固体
密度
1.98g/cm3
熔点
158-160ºC
折射率
1.896