化合物简介
Eletriptan (trade name Relpax, used in the form of eletriptan hydrobromide) is a second generation triptan drug intended for treatment of migraine headaches. It is used as an abortive medication, blocking a migraine attack which is already in progress. Eletriptan is marketed and manufactured by Pfizer Inc. It is sold in the US and Canada under the brand name Relpax, and in several other countries under the brand name Relert.
基本信息
中文名称
依来曲普坦
英文名称
eletriptan
中文别名
氢溴酸依利曲坦、3-苄基-5-(1-(2-(吡咯烷-1-基)乙基)-1H-吲哚-3-基)-1,2,4-恶二唑、3-[(1-甲基吡咯烷-2-基)甲基]-5-(2-苯基磺酰乙基)-1H-吲哚
英文别名
Eletriptan、5-[2-(benzenesulfonyl)ethyl]-3-[[(2R)-1-methylpyrrolidin-2-yl]methyl]-1H-indole
CAS号
143322-58-1
分子式
C22H26N2O2S
分子量
382.519
精确质量
382.171
PSA
61.55
LOGP
4.8397
物化性质
外观与性状
黄色泡沫
密度
1.235 g/cm3
沸点
613.4ºC at 760 mmHg
闪点
324.8ºC
蒸汽压
1.58E-16mmHg at 25°C
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